Cerestat is a potent and noncompetitive NMDA receptor antagonist (IC50 = 36 nM). Exhibits >70-fold selectivity for NMDA receptor over σ receptor. Neuroprotective in a rat model of focal ischemia.
- Nom chimique ou matériau
- Cerestat
- CAS
- 137160-11-3
- Synonyme
- N-(3-Ethylphenyl)-N-methyl-N'-1-naphthalenylguanidine hydrochloride
- Quantité
- 50 mg
- Solubilité
- Soluble to 50mM in water and to 100mM in DMSO
- Formule moléculaire
- C20H21N3·HCl
- Poids de la formule
- 339.86
- Forme physique
- Solid
- Type de produit
- Bioactive Small Molecule
- Pureté
- >98%
