193 D7 is a histone demethylase JMJD1C inhibitor (IC50 = 0.59 μM in in vitro demethylation assay). In vivo, 193 D7 suppresses tumor by targeting intratumoral Treg cells in mice tumor models. 193 D7 is orally bioavailable.
- Nom chimique ou matériau
- 8-Benzoyl-2,3,6,7-tetrahydro-5-oxo-5H-thiazolo[3,2-a]pyridine-6-acetic acid
- CAS
- 861224-48-8
- Quantité
- 50 mg
- Cible
- Histone Demethylase Inhibitors
- Formule moléculaire
- C16H15NO4S
- Pureté
- 0.98