Potent GnRH receptor antagonist
Cetrorelix acetate is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist (KD = 0.202 nM, IC50 = 1.21 nM). Suppresses production of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland, which inhibits ovulation. Exhibits antiproliferative effects and displays efficacy against hormone-sensitive cancers
in vivo
. Also exhibits anxiolytic and antidepressant activity
in vivo
| Marque | Tocris Bioscience |
|---|---|
| Réf. B-LABO | BL-RE-178196 |
| Réf. fabricant | 30306094 |
| CAS | 145672-81-7 |
| Quantité | 1 mg |
| Cible | GnRH Antagonist |
| Formule moléculaire | C70H92ClN17O14 |
| Pureté | 0.95 |
