Cetrorelix acetate is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist (KD = 0.202 nM, IC50 = 1.21 nM). Suppresses production of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland, which inhibits ovulation. Exhibits antiproliferative effects and displays efficacy against hormone-sensitive cancers in vivo. Also exhibits anxiolytic and antidepressant activity in vivo.
- CAS
- 145672-81-7
- Quantité
- 1 mg
- Cible
- GnRH Antagonist
- Formule moléculaire
- C70H92ClN17O14
- Pureté
- 0.95
