AF 64394 is a potent and selective GPR3 inverse agonist (pIC50 = 7.3). Selective for GPR3 over GPR6 and GPR12 (pIC50 values are 5.1 and 4.9, respectively).
- Nom chimique ou matériau
- N-[[4-Chloro-2-(1-methylethoxy)phenyl]methyl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
- CAS
- 1637300-25-4
- Quantité
- 50 mg
- Formule moléculaire
- C21H20ClN5O
- Pureté
- 98%