DY 268 is a potent FXR antagonist (IC50 = 7.5 nM). Exhibits no detectable cytotoxicity in cell-based assays.
- Nom chimique ou matériau
- 1-[(3-Methoxyphenyl)methyl]-N-[4-methyl-3-(4-morpholinylsulfonyl)phenyl]-3-(4-methylphenyl)-1H-pyrazole-4-carboxamide
- CAS
- 1609564-75-1
- Quantité
- 50 mg
- Cible
- LXR-like Receptor Antagonists
- Formule moléculaire
- C30H32N4O5S
- Poids de la formule
- 560.66
- Pureté
- >98%