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Tocris Bioscience™ ERK5-IN-1

Name: Tocris Bioscience™ ERK5-IN-1
Brand: Tocris Bioscience
SKU: 18747068
Price: 350.96 EUR
Availability: InStock

Réf. : BL-RE-142997Réf. fabricant : 18747068 10 mg

350,96 € HT

Potent and selective ERK5 inhibitor

Pureté: >98%
Description: ERK5-IN-1
Poids moléculaire: 638.8
Type de produit: ERK5-IN-1
Quantité: 10 mg
Marque: Tocris Bioscience

ERK5-IN-1 is a potent and selective ERK5 inhibitor; inhibits EGFR-induced ERK5 autophosphorylation (EC50 = 90 nM) and ERK5 enzymatic activity (IC50 = 162 nM). Exhibits at least 30-fold selectivity for ERK5 over LRRK2 in a cell based assay. Also selective for ERK5 over a panel of other kinases. Orally bioavailable.