Tocris Bioscience™ AY 77

Ref : 18709956
362.84

Potent PAR2 biased agonist; exhibits bias for Ca2+ signaling

Pureté :
95%
CAS :
1835734-92-3
Contenu et stockage :
Store at -20°C
Poids moléculaire :
M.W.-observed: 404.5
Quantité :
1 mg
Brand
Tocris Bioscience™

AY 77 is a potent PAR2 biased agonist. AY 77 exhibits bias for Ca2+ over ERK1/2 signaling (EC50 values are 40 nM for Ca2+ release versus 2 μM for ERK1/2 phosphorylation). Shows selectivity for PAR2 over PAR1. Promotes migration of human breast cancer cells in vitro.

Pureté : 95%


CAS : 1835734-92-3


Contenu et stockage : Store at -20°C


Poids moléculaire : M.W.-observed: 404.5


Quantité : 1 mg