Tocris Bioscience™ MS 143
348,80 € HT
AKT kinase Degrader (PROTAC™)
- Marque
- Tocris Bioscience
"/>
AKT kinase Degrader (PROTAC™)
MS 143 is a potent and selective protein kinase B (AKT) Degrader (PROTAC™) (DC50 = 46 nM, Dmax = 100 % at 24h in PC3 cells). MS 143 suppresses growth in prostate cancer PC3 cells; suppresses tumor growth and reduces AKT protein levels in a mouse PC3 cell xenograft model.
PROTAC™ is a registered trademark of Arvinas Operations, Inc., and is used under license.
| Marque | Tocris Bioscience |
|---|---|
| Réf. B-LABO | BL-RE-177672 |
| Réf. fabricant | 30279883 |