CYN 154806 is a potent and selective somatostatin sst2 receptor antagonist. pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively.
- Pureté
- 0.95
- Contenu et stockage
- Store at -20°C
- Description
- CYN 154806
- Poids moléculaire
- 1197.35
- Type de produit
- CYN 154806
- Quantité
- 1 mg
- Séquence
- Ac-(4-Nitro)Phe-D-Cys-Tyr-D-Trp-Lys-Thr-Cys-D-Tyr-NH2 (Disulfide bridge: 2 - 7)