PBP 10 is a selective formyl peptide receptor 2 (FPR2) antagonist; cell permeable. Selectively inhibits FPR2-mediated NADPH oxidase activity but has no effect on FPR1 signaling in neutrophils. Displays PIP2 binding activity
in vitro
and blocks cell motility. Also exhibits antiviral activity against influenza viruses via inhibition of viral-induced ERK activation.
Caractéristiques techniques
| Marque | Tocris Bioscience |
| Réf. B-LABO | BL-RE-055936 |
| Réf. fabricant | 18755727 |
| Pureté | 95% |
|---|
| Contenu et stockage | Store at -20°C |
|---|
| Poids moléculaire | M.W. (Observed): 1712.1 |
|---|
| Quantité | 1 mg |
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